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S. Creason

Journal of Medicinal Chemistry, ACS Applied Materials and Interfaces, Biomaterials, European journal of medicinal chemistry, Antimicrobial Agents and Chemotherapy
9
Role
Title
Level Year L/R
🐜 Identification of a metabolically stable triazolopyrimidine-based dihydroorotate dehydrogenase inhibitor with antimalarial activity in mice.
13 auth. R. Gujjar, A. Marwaha, Farah El Mazouni, John White, K. White, S. Creason, David M. Shackleford, J. Baldwin, W. Charman, F. Buckner, ... S. Charman, P. Rathod, M. Phillips 		7 2009
7
🐜
🐜 Lead optimization of aryl and aralkyl amine-based triazolopyrimidine inhibitors of Plasmodium falciparum dihydroorotate dehydrogenase with antimalarial activity in mice.
16 auth. R. Gujjar, Farah El Mazouni, K. White, John White, S. Creason, David M. Shackleford, Xiao-Yi Deng, W. Charman, I. Bathurst, J. Burrows, ... D. Floyd, D. Matthews, F. Buckner, S. Charman, M. Phillips, P. Rathod 		7 2011
7
🐜
🐜 Bioisosteric transformations and permutations in the triazolopyrimidine scaffold to identify the minimum pharmacophore required for inhibitory activity against Plasmodium falciparum dihydroorotate dehydrogenase.
9 auth. A. Marwaha, John White, Farah El Mazouni, S. Creason, Sreekanth Kokkonda, F. Buckner, ... S. Charman, M. Phillips, P. Rathod 		5 2012
5
🐜
🐜 Substituted 2-phenylimidazopyridines: a new class of drug leads for human African trypanosomiasis.
18 auth. H. Tatipaka, J. R. Gillespie, A. Chatterjee, Neil R. Norcross, Matthew A. Hulverson, Ranae M. Ranade, P. Nagendar, S. Creason, J. McQueen, Nicole A Duster, ... A. Nagle, F. Supek, V. Molteni, T. Wenzler, R. Brun, R. Glynne, F. Buckner, M. Gelb 		5 2014
5
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🐜 Urea Derivatives of 2-Aryl-benzothiazol-5-amines: A New Class of Potential Drugs for Human African Trypanosomiasis.
10 auth. D. A. Patrick, J. Gillespie, J. McQueen, Matthew A. Hulverson, Ranae M. Ranade, S. Creason, ... Zackary M Herbst, Michael H. Gelb, F. Buckner, R. Tidwell 		5 2017
5
🐜
🐜 Photoreactive Carboxybetaine Copolymers Impart Biocompatibility and Inhibit Plasticizer Leaching on Polyvinyl Chloride.
11 auth. Xiaojie Lin, Kan Wu, Qiong Zhou, Priyesh Jain, Mary O'Kelly Boit, Bowen Li, ... Hsiang-Chieh Hung, S. Creason, J. Himmelfarb, B. Ratner, Shaoyi Jiang 		5 2020
5
🐜
🐜 Precision-porous polyurethane elastomers engineered for application in pro-healing vascular grafts: Synthesis, fabrication and detailed biocompatibility assessment.
9 auth. Le Zhen, S. Creason, Felix I. Simonovsky, J. Snyder, Sarah L. Lindhartsen, Marvin Mecwan, ... Brian W. Johnson, J. Himmelfarb, B. Ratner 		4 2021
4
🐜
🐜 Structure-guided design of novel Trypanosoma brucei Methionyl-tRNA synthetase inhibitors.
12 auth. Wenlin Huang, Zhongsheng Zhang, X. Barros-Álvarez, C. Koh, Ranae M. Ranade, J. R. Gillespie, ... S. Creason, S. Shibata, C. Verlinde, W. Hol, F. Buckner, E. Fan 		4 2016
4
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🐜 Development of Methionyl-tRNA Synthetase Inhibitors as Antibiotics for Gram-Positive Bacterial Infections
12 auth. O. Faghih, Zhongsheng Zhang, Ranae M. Ranade, J. R. Gillespie, S. Creason, Wenlin Huang, ... S. Shibata, X. Barros-Álvarez, C. Verlinde, Wim G. J. Hol, E. Fan, F. Buckner 		4 2017
4
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