π
|
Design, Synthesis and Evaluation of New Quinazolinone Derivatives that Inhibit Bloom's Syndrome Protein (BLM) Helicase, Trigger DNA damage at the Telomere Region and Synergize with PARP Inhibitors.
15 auth.
Chen-Xi Wang,
Zi-Lin Zhang,
Qi-Kun Yin,
Jia-Li Tu,
Jia-En Wang,
Yao-Hao Xu,
Yong Rao,
Tian-Miao Ou,
Shi-Liang Huang,
Ding Li,
...
Honggen Wang,
Qingjiang Li,
Jia-Heng Tan,
Shuo-Bin Chen,
Zhishu Huang
|
4 |
2020 |
4 π
|
π
|
A novel HSF1 activator ameliorates nonβalcoholic steatohepatitis by stimulating mitochondrial adaptive oxidation
16 auth.
Yong Rao,
Chan Li,
Yu-Tao Hu,
Yao-Hao Xu,
Bing-Bing Song,
Shiying Guo,
Zhiyuan Jiang,
Dandan Zhao,
Shuo-Bin Chen,
Jia-Heng Tan,
...
Shi-Liang Huang,
Qingjiang Li,
Xiao-Jun Wang,
Ying-jun Zhang,
JiβMing Ye,
Zhishu Huang
|
3 |
2021 |
3 π
|
π
|
Design, Synthesis, and Evaluation of New Sugar-Substituted Imidazole Derivatives as Selective c-MYC Transcription Repressors Targeting the Promoter G-Quadruplex.
12 auth.
Mao-lin Li,
Jing-Mei Yuan,
Haoxuan Yuan,
Bi-Han Wu,
Shi-Liang Huang,
Qingjiang Li,
...
Tian-Miao Ou,
Honggen Wang,
Jia-Heng Tan,
Ding Li,
Shuo-Bin Chen,
Zhishu Huang
|
3 |
2022 |
3 π
|
π
|
Discovery of a promising agent IQZ23 for the treatment of obesity and related metabolic disorders.
17 auth.
Yong Rao,
Zhao Xu,
Yu-Tao Hu,
Chan Li,
Yao-Hao Xu,
Qin-Qin Song,
Hong Yu,
Bing-Bing Song,
Shuo-Bin Chen,
Qingjiang Li,
...
Shi-Liang Huang,
Jia-Heng Tan,
Tian-Miao Ou,
Honggen Wang,
G. Zhong,
JiβMing Ye,
Zhishu Huang
|
3 |
2020 |
3 π
|
π
|
Discovery of a Novel G-Quadruplex and Histone Deacetylase (HDAC) Dual-Targeting Agent for the Treatment of Triple-Negative Breast Cancer.
14 auth.
Xingpeng Jiang,
Fang-Hai Tu,
Li-Yuan Wei,
Bo Wang,
Hao Yuan,
Jing-Mei Yuan,
Yong Rao,
Shi-Liang Huang,
Qingjiang Li,
Tian-Miao Ou,
...
Honggen Wang,
Jia-Heng Tan,
Shuo-Bin Chen,
Zhishu Huang
|
3 |
2022 |
3 π
|
π
|
Design and Synthesis of Bouchardatine Derivatives as a Novel AMP-Activated Protein Kinase Activator for the Treatment of Colorectal Cancer.
15 auth.
Yao-Hao Xu,
Yu-Tao Hu,
Shu-Min Xu,
Bing-Bing Song,
Haonan Yuan,
Dan-Dan Zhao,
ShiβYao Guo,
Zhiyuan Jiang,
Li-Yuan Wei,
Yong Rao,
...
Jia-Heng Tan,
Shi-Liang Huang,
Qingjiang Li,
Shuo-Bin Chen,
Z. Huang
|
2 |
2023 |
2 π
|