π
|
A small molecule that induces translational readthrough of CFTR nonsense mutations by eRF1 depletion
30 auth.
Jyoti Sharma,
M. Du,
E. Wong,
V. Mutyam,
Yao Li,
Jianguo Chen,
J. Wangen,
Kari Thrasher,
Lianwu Fu,
N. Peng,
L. Tang,
Kaimao Liu,
Bini Mathew,
R. Bostwick,
C. Augelli-Szafran,
...
H. Bihler,
F. Liang,
J. Mahiou,
J. Saltz,
A. Rab,
Jeong-Soo Hong,
E. Sorscher,
E. Mendenhall,
Candice J. Coppola,
K. Keeling,
R. Green,
M. Mense,
M. Suto,
S. Rowe,
D. Bedwell
|
6 |
2021 |
6 π
|
π
|
Identification of an Anti-diabetic, Orally Available Small Molecule that Regulates TXNIP Expression and Glucagon Action.
15 auth.
L. Thielen,
Junqin Chen,
Gu Jing,
O. Moukha-Chafiq,
Guanlan Xu,
Seongho Jo,
T. Grayson,
Brian Lu,
Peng Li,
C. Augelli-Szafran,
...
M. Suto,
Matt Kanke,
P. Sethupathy,
Jason K. Kim,
A. Shalev
|
5 |
2020 |
5 π
|
π
|
The G2019S mutation in LRRK2 imparts resiliency to kinase inhibition
7 auth.
Kaela Kelly,
Shijie Wang,
Ravindra Boddu,
Zhiyong Liu,
O. Moukha-Chafiq,
C. Augelli-Szafran,
...
A. West
|
5 |
2018 |
5 π
|
π
|
Preferential Inhibition of Wnt/Ξ²-Catenin Signaling by Novel Benzimidazole Compounds in Triple-Negative Breast Cancer
7 auth.
Abhishek Gangrade,
V. Pathak,
C. Augelli-Szafran,
Han-Xun Wei,
P. Oliver,
M. Suto,
...
D. Buchsbaum
|
5 |
2018 |
5 π
|
π
|
Discovery of a novel inhibitor of kinesin-like protein KIFC1.
17 auth.
Wei Zhang,
L. Zhai,
Yimin Wang,
R. Boohaker,
Wenyan Lu,
Vandana Gupta,
I. Padmalayam,
R. Bostwick,
E. White,
L. Ross,
...
J. Maddry,
S. Ananthan,
C. Augelli-Szafran,
M. Suto,
Bo Xu,
Rongbao Li,
Yonghe Li
|
5 |
2016 |
5 π
|
π
|
Regulation of Tumor Immunity by Lysophosphatidic Acid
7 auth.
Suechin Lee,
MΓ©lanie A. Dacheux,
Derek D Norman,
L. BalΓ‘zs,
R. Torres,
C. Augelli-Szafran,
...
G. Tigyi
|
4 |
2020 |
4 π
|
π
|
Pyrimidone inhibitors targeting Chikungunya Virus nsP3 macrodomain by fragment-based drug design
11 auth.
Sixue Zhang,
A. Garzan,
Nicole N Haese,
R. Bostwick,
Yohanka Martinez-Gzegozewska,
L. Rasmussen,
...
D. Streblow,
Mark T Haise,
A. Pathak,
C. Augelli-Szafran,
Mousheng Wu
|
4 |
2021 |
4 π
|
π
|
Identification of Compounds That Decrease Glioblastoma Growth and Glucose Uptake in Vitro.
14 auth.
Catherine J. Libby,
Sixue Zhang,
G. Benavides,
Sarah E. Scott,
Yanjie Li,
M. Redmann,
A. Tran,
Arphaxad Otamias,
V. Darley-Usmar,
M. Napierala,
...
Jianhua Zhang,
C. Augelli-Szafran,
Wei Zhang,
A. Hjelmeland
|
4 |
2018 |
4 π
|