|
🐜
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Cyclin-dependent kinase 12, a novel drug target for visceral leishmaniasis
32 auth.
S. Wyllie,
Michael G. Thomas,
Stephen Patterson,
Sabrinia D Crouch,
M. De Rycker,
R. Lowe,
S. Gresham,
Michael D. Urbaniak,
T. Otto,
L. Stojanovski,
Frederick R. C. Simeons,
Sujatha Manthri,
Lorna M MacLean,
F. Zuccotto,
Nadine Homeyer,
...
H. Pflaumer,
Markus Boesche,
Lalitha Sastry,
P. Connolly,
S. Albrecht,
M. Berriman,
G. Drewes,
David W. Gray,
S. Ghidelli-Disse,
S. Dixon,
J. Fiandor,
P. Wyatt,
M. Ferguson,
A. Fairlamb,
T. Miles,
K. Read,
I. Gilbert
|
6 |
2018 |
6
🐜
|
|
🐜
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Synthesis, antimalarial activity, and preclinical pharmacology of a novel series of 4'-fluoro and 4'-chloro analogues of amodiaquine. Identification of a suitable "back-up" compound for N-tert-butyl isoquine.
29 auth.
P. O’Neill,
A. Shone,
Deborah Stanford,
G. Nixon,
E. Asadollahy,
B. Park,
J. Maggs,
P. Roberts,
Paul A. Stocks,
G. Biagini,
P. Bray,
Jill Davies,
N. Berry,
Charlotte Hall,
Karen Rimmer,
...
P. Winstanley,
S. Hindley,
R. Bambal,
C. Davis,
M. Bates,
S. Gresham,
R. Brigandi,
Federico M Gomez-de-Las-Heras,
D. Gargallo,
S. Parapini,
L. Vivas,
H. Lander,
D. Taramelli,
S. Ward
|
5 |
2009 |
5
🐜
|
|
🐜
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First-Time-in-Human Study and Prediction of Early Bactericidal Activity for GSK3036656, a Potent Leucyl-tRNA Synthetase Inhibitor for Tuberculosis Treatment
14 auth.
D. Tenero,
G. Derimanov,
Alex Carlton,
J. Tonkyn,
M. Davies,
S. Cozens,
S. Gresham,
A. Gaudion,
Adeep Puri,
M. Muliaditan,
...
Joaquin Rullas-Trincado,
Alfonso Mendoza-Losana,
A. Skingsley,
David Barros-Aguirre
|
5 |
2019 |
5
🐜
|
|
🐜
|
Identification of GSK3186899/DDD853651 as a Preclinical Development Candidate for the Treatment of Visceral Leishmaniasis
52 auth.
Michael G. Thomas,
M. De Rycker,
M. Ajakane,
S. Albrecht,
A. Álvarez-Pedraglio,
Markus Boesche,
S. Brand,
Lorna Campbell,
Juan Cantizani-Perez,
Laura A. T. Cleghorn,
R. Copley,
Sabrinia D Crouch,
A. Daugan,
G. Drewes,
S. Ferrer,
...
S. Ghidelli-Disse,
Silvia González,
S. Gresham,
A. Hill,
S. Hindley,
R. Lowe,
Claire J. Mackenzie,
Lorna M MacLean,
Sujatha Manthri,
Franck Martin,
Juan Miguel-Siles,
Van-Loc Nguyen,
S. Norval,
Maria Osuna-Cabello,
Andrew Woodland,
Stephen Patterson,
Imanol Peña,
Maria Teresa Quesada-Campos,
Iain H Reid,
Charlotte H. Revill,
Jennifer Riley,
J. Ruiz-Gomez,
Y. Shishikura,
Frederick R. C. Simeons,
Alasdair R C Smith,
V. Smith,
D. Spinks,
L. Stojanovski,
John Thomas,
S. Thompson,
Tim Underwood,
David W. Gray,
J. Fiandor,
I. Gilbert,
P. Wyatt,
K. Read,
T. Miles
|
5 |
2018 |
5
🐜
|
|
🐜
|
The small-molecule SMARt751 reverses Mycobacterium tuberculosis resistance to ethionamide in acute and chronic mouse models of tuberculosis
41 auth.
Marion Flipo,
Rosangela Frita,
M. Bourotte,
María S Martínez-Martínez,
Markus Boesche,
G. Boyle,
G. Derimanov,
G. Drewes,
Pablo Gamallo,
S. Ghidelli-Disse,
S. Gresham,
E. Jiménez,
Jaime de Mercado,
Esther Pérez-Herrán,
Esther Porras-De Francisco,
...
J. Rullas,
Patricia Casado,
F. Leroux,
Catherine Piveteau,
Mehdi Kiass,
V. Mathys,
K. Soetaert,
Véronique Megalizzi,
A. Tanina,
R. Wintjens,
R. Antoine,
P. Brodin,
V. Delorme,
M. Moune,
Kamel Djaout,
S. Slupek,
C. Kemmer,
M. Gitzinger,
Lluís Ballell,
Alfonso Mendoza-Losana,
S. Lociuro,
B. Déprez,
David Barros-Aguirre,
M. Remuiñán,
N. Willand,
A. Baulard
|
4 |
2022 |
4
🐜
|
|
🐜
|
Author Correction: Cyclin-dependent kinase 12 is a drug target for visceral leishmaniasis
32 auth.
S. Wyllie,
Michael G. Thomas,
Stephen Patterson,
Sabrinia D Crouch,
M. Rycker,
R. Lowe,
S. Gresham,
Michael D. Urbaniak,
T. Otto,
L. Stojanovski,
Frederick R. C. Simeons,
Sujatha Manthri,
Lorna M MacLean,
F. Zuccotto,
Nadine Homeyer,
...
H. Pflaumer,
Markus Boesche,
Lalitha Sastry,
Paul Connolly,
S. Albrecht,
M. Berriman,
G. Drewes,
David W. Gray,
S. Ghidelli-Disse,
S. Dixon,
J. Fiandor,
P. Wyatt,
Michael A J Ferguson,
A. Fairlamb,
T. Miles,
K. Read,
I. Gilbert
|
3 |
2023 |
3
🐜
|
|
🐜
|
A human microdose study of the antimalarial drug GSK3191607 in healthy volunteers
15 auth.
Malek Okour,
G. Derimanov,
Rodger Barnett,
Esther Fernández,
S. Ferrer,
S. Gresham,
Mohammad Hossain,
F. Gamo,
G. Koh,
Adrian I. Pereira,
...
K. Rolfe,
Deborah Wong,
G. Young,
H. Rami,
J. Haselden
|
3 |
2018 |
3
🐜
|
|
🐬
|
Comparative embryotoxicity of diverse anti-malarial compounds using rat whole embryo culture and the application of the screen in lead identification for diseases of the developing world molecules
A. James,
J. Haselden,
S. Gresham,
Pablo Castañeda-Casado,
E. Jimenez-Navarro,
P. Bushdid
|
0 |
2014 |
0
🐬
|
